SCHEMBL28848874

SCHEMBL28848874

COc1cnc(NC(=O)OC(C)(C)C)cc1-n1cnc(C2CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
MAP3K5 Q99683 17/20 0.41
AKT1 P31749 5/20 0.37
TGFBR1 P36897 1/20 0.37
MAPKAPK2 P49137 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28848741 0.88 MAP3K5 (0.46) GSK3BDYRK1AMAP3K5
SCHEMBL29949315 0.78 MAP3K5 (0.43) MAP3K5AKT1
SCHEMBL28648080 0.78 MAP3K5 (0.43) MAP3K5AKT1
SCHEMBL28658716 0.76 MAP3K5 (0.41) MAP3K5AKT1
SCHEMBL29949144 0.76 MAP3K5 (0.41) MAP3K5AKT1
SCHEMBL28663432 0.76 MAP3K5 (0.41) MAP3K5AKT1
SCHEMBL16692819 0.76 PSEN1 (0.44) GSK3BDYRK1A
Hydrochloric Acid SCHEMBL28656984 0.76 MAP3K5 (0.41) MAP3K5AKT1
SCHEMBL28660361 0.76 MAP3K5 (0.43) MAP3K5AKT1
SCHEMBL28848835 0.75 MAP3K5 (0.45) MAP3K5TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110036005-B Amide derivatives and their use in medicine 广东东阳光药业有限公司 2022-09-27 CN disclosed