SCHEMBL28849680

SCHEMBL28849680

COc1ccc(-c2c(N)n[nH]c2OC)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
DYRK1A Q13627 1/20 0.51
MAPT P10636 4/20 0.47
RAB9A P51151 2/20 0.46
GAA P10253 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HEXA P06865 1/20 0.46
HEXB P07686 1/20 0.46
GFER P55789 1/20 0.46
HTT P42858 1/20 0.46
MAPK10 P53779 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
IKBKB O14920 2/20 0.45
MAP3K14 Q99558 1/20 0.45
NPC1 O15118 1/20 0.45
MAPK1 P28482 1/20 0.45
CHUK O15111 1/20 0.45
IKBKE Q14164 1/20 0.44
LMNA P02545 1/20 0.44
APP P05067 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28171296 0.86 AKT2 (0.61) KDM4EALDH1A1IKBKBMAP3K14MAPK1
SCHEMBL13312276 0.82 IKBKB (0.67) KDM4EDYRK1AGAAALDH1A1IKBKB
SCHEMBL17731310 0.77 HTT (0.48) KDM4EDYRK1AMAPTRAB9AGAA
SCHEMBL8034982 0.75 HTT (0.56) KDM4EDYRK1AMAPTRAB9AGAA
SCHEMBL13516427 0.74 MAPT (0.50) KDM4EDYRK1AMAPTRAB9AGAA
SCHEMBL28067319 0.74 MAPT (0.50) KDM4EDYRK1AMAPTRAB9AGAA
SCHEMBL8097613 0.72 TDP1 (0.56) KDM4EDYRK1AMAPTRAB9AALDH1A1
SCHEMBL3364101 0.71 JAK2 (0.66) DYRK1ACHUK
SCHEMBL12907168 0.71 PRKAG1 (0.68) DYRK1A
SCHEMBL4898151 0.71 KDM4E (0.51) KDM4EDYRK1AMAPTRAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107108638-A Piperidyl PyrazolopyrimidinonecGMP and application thereof 拜耳制药股份公司 2017-08-29 CN disclosed