SCHEMBL28853802

SCHEMBL28853802

COc1ccc(C(CS(C)(=O)=O)C2C=CCS2)cc1OCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.42
PDE4A P27815 4/20 0.42
PDE4C Q08493 4/20 0.42
PDE4D Q08499 4/20 0.42
SMPD1 P17405 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ACHE P22303 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28189250 0.89 PDE4B (0.39) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL28189206 0.89 PDE4B (0.39) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL28853800 0.88 PDE4B (0.48) PDE4BPDE4APDE4CPDE4D
SCHEMBL28189207 0.88 PDE4B (0.48) PDE4BPDE4APDE4CPDE4D
SCHEMBL28853737 0.88 PDE4B (0.48) PDE4BPDE4APDE4CPDE4D
SCHEMBL4371698 0.78 MEN1 (0.44) MEN1KMT2APOLBGAAF2
SCHEMBL4366818 0.77 APP (0.40) MEN1KMT2APOLBGAAF2
SCHEMBL9938952 0.77 PDE4A (0.48) PDE4BPDE4APDE4CPDE4DSMPD1
SCHEMBL4372450 0.76 MEN1 (0.48) MEN1KMT2AGAAMAPK1APP
SCHEMBL4369067 0.75 APP (0.53) MEN1KMT2APOLBGAAAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108059635-A Thiophene derivant 天津合美医药科技有限公司 2018-05-22 CN claimed
CN-107964016-A Thiophene derivant 天津合美医药科技有限公司 2018-04-27 CN claimed
CN-107722036-A Thiophene derivant 天津合美医药科技有限公司 2018-02-23 CN claimed
CN-107501290-A Thiophene derivant 天津合美医药科技有限公司 2017-12-22 CN claimed
CN-108059635-A Thiophene derivant 天津合美医药科技有限公司 2018-05-22 CN disclosed
CN-107964016-A Thiophene derivant 天津合美医药科技有限公司 2018-04-27 CN disclosed
CN-107722036-A Thiophene derivant 天津合美医药科技有限公司 2018-02-23 CN disclosed
CN-107501290-A Thiophene derivant 天津合美医药科技有限公司 2017-12-22 CN disclosed