Phenyltoloxamine

Phenyltoloxamine

SCHEMBL28854

CN(C)CCOc1ccccc1Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 1.00
DRD2 P14416 2/20 1.00
DRD4 P21917 2/20 1.00
DRD5 P21918 2/20 1.00
HRH1 P35367 5/20 0.85
DRD3 P35462 2/20 0.72
LMNA P02545 2/20 0.70
KDM4E B2RXH2 1/20 0.70
HPGD P15428 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
LTA4H P09960 1/20 0.61
TP53 P04637 1/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2C9 P11712 1/20 0.60
TSHR P16473 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
HTR7 P34969 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenyltoloxamine SCHEMBL5145512 1.00 DRD1 (1.00) DRD1DRD2DRD4DRD5HRH1
Phenyltoloxamine SCHEMBL16755246 0.98 DRD1 (0.97) DRD1DRD2DRD4DRD5HRH1
SCHEMBL11754849 0.92 HRH1 (1.00) DRD1DRD2DRD4DRD5HRH1
SCHEMBL10989007 0.90 HRH1 (0.91) DRD1DRD2DRD4DRD5HRH1
Hydrochloric Acid SCHEMBL11629488 0.89 HRH1 (0.88) DRD1DRD2DRD4DRD5HRH1
Phenyltoloxamine SCHEMBL8510190 0.89 HRH1 (1.00) DRD1DRD2DRD4DRD5HRH1
Diphenhydramine SCHEMBL8036949 0.88 DRD1 (0.77) DRD1DRD2DRD4DRD5HRH1
Diphenhydramine SCHEMBL8040055 0.88 DRD1 (0.77) DRD1DRD2DRD4DRD5HRH1
SCHEMBL10800339 0.88 DRD2 (0.78) DRD1DRD2DRD4DRD5HRH1
SCHEMBL10768290 0.88 DRD2 (0.78) DRD1DRD2DRD4DRD5HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5680 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4731194-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP Technologies, Inc. (US) 2026-04-29 EP claimed
WO-2025264260-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP TECHNOLOGIES, INC. (US) 2025-12-26 WO claimed
EP-4630401-A2 CARBONIC ANHYDRASE ENZYME INHIBITORS AND METHODS OF USE THEREOF Rutgers, the State University of New Jersey (US) 2025-10-15 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-20250177398-A1 CARBONIC ANHYDRASE ENZYMES FOR REGULATING MAST CELL HEMATOPOIESIS AND TYPE 2 INFLAMMATION RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2025-06-05 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
US-12263168-B2 Carbonic anhydrase enzymes for regulating mast cell hematopoiesis and type 2 inflammation RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2025-04-01 US claimed
US-20250099498-A1 STRONTIUM BASED COMPOSITIONS AND FORMULATIONS FOR PAIN, PRURITUS, AND INFLAMMATION GALLEON LABS LLC (US) 2025-03-27 US claimed
US-12251469-B2 Sterically stabilized carrier compositions for treating a mammal VGSK TECHNOLOGIES, INC. (US) 2025-03-18 US claimed
EP-0132472-B1 MEDICATED PRODUCTS CONTAINING A MAGNESIUM TRISILICATE ADSORBENT WITH A MEDICAMENT DRUG ADSORBED THEREON WARNER-LAMBERT COMPANY (US) 1989-06-21 EP claimed
US-4753800-A DRUGS ADSORBED ONTO MAGNESIUM ALUMINUM STEARATE WARNER-LAMBERT COMPANY (US) 1988-06-28 US claimed
US-4749700-A NASAL ADMINISTRATION LOWER DOSAGE NASTECH PHARMACEUTICAL CO, INC. (US) 1988-06-07 US claimed
EP-0219458-A2 Medicament adsorbates and their preparation WARNER-LAMBERT COMPANY (US) 1987-04-22 EP claimed
US-4642231-A Magnesium trisilicate suitable for preparation of medicament adsorbates of antihistamines WARNER-LAMBERT COMPANY (US) 1987-02-10 US claimed
EP-0180597-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS. SUNSHINE ABRAHAM (US) 1986-05-14 EP claimed
WO-1985004589-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS SUNSHINE ABRAHAM 1985-10-24 WO claimed
EP-0132472-A1 Medicated products containing a magnesium trisilicate adsorbent with a medicament drug adsorbed thereon WARNER-LAMBERT COMPANY (US) 1985-02-13 EP claimed
US-4104382-A (((THIAZOLYL-, ISOTHIAZOLYL- OR PYRIDYLALKYL)THIO)ALKYL)GUANIDINE SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1978-08-01 US claimed
US-4000302-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1976-12-28 US claimed