SCHEMBL28863201

SCHEMBL28863201

Nc1ccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)cn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 11/20 1.00
CDK7 P50613 2/20 0.69
CDK6 Q00534 2/20 0.69
KDR P35968 6/20 0.67
RAF1 P04049 4/20 0.67
BRAF P15056 2/20 0.63
PDGFRB P09619 2/20 0.62
KIT P10721 2/20 0.62
PDGFRA P16234 2/20 0.62
FGFR2 P21802 2/20 0.62
FLT3 P36888 2/20 0.62
CA7 P43166 2/20 0.62
CA9 Q16790 2/20 0.62
MEN1 O00255 1/20 0.62
PLK4 O00444 1/20 0.62
CIT O14578 1/20 0.62
AURKA O14965 1/20 0.62
MUSK O15146 1/20 0.62
EPHB6 O15197 1/20 0.62
MAPK13 O15264 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29996391 0.92 CDK8 (1.00) CDK8CDK7CDK6RETCCNC
SCHEMBL28863217 0.92 CDK8 (1.00) CDK8CDK7CDK6RETCCNC
SCHEMBL28863252 0.88 CDK8 (1.00) CDK8CDK7CDK6KDRBRAF
SCHEMBL28863218 0.86 CDK8 (0.83) CDK8CDK7CDK6CA9EPHX2
SCHEMBL4344749 0.86 RAF1 (0.78) CDK8CDK7CDK6KDRRAF1
SCHEMBL5899269 0.85 CDK8 (0.74) CDK8CDK7CDK6KDRRAF1
SCHEMBL620425 0.84 RAF1 (0.79) CDK8CDK7CDK6KDRRAF1
SCHEMBL619479 0.84 CDK8 (0.73) CDK8CDK7CDK6KDRRAF1
SCHEMBL28863221 0.83 CDK8 (0.84) CDK8CDK7CDK6MEN1KMT2A
SCHEMBL3174505 0.83 CDK8 (0.71) CDK8CDK7CDK6KDRRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115197130-B Aryl urea derivative and preparation method and application thereof 安徽医科大学 2023-06-27 CN disclosed
CN-115197130-A Aryl urea derivative and preparation method and application thereof 安徽医科大学 2022-10-18 CN disclosed