SCHEMBL28865440

SCHEMBL28865440

Brc1cccc(C2(Nc3ncccn3)CCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 16/20 0.46
HDAC3 O15379 15/20 0.46
HDAC1 Q13547 15/20 0.46
HDAC2 Q92769 15/20 0.46
VNN1 O95497 2/20 0.40
GPR39 O43194 1/20 0.38
CTSD P07339 1/20 0.37
BACE1 P56817 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24968663 0.86 HDAC3 (0.53) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28247580 0.83 HDAC6 (0.49) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL30145542 0.82 HDAC6 (0.62) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28248201 0.82 HDAC6 (0.62) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28247582 0.80 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28248177 0.78 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28248169 0.78 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL1030969 0.78 HDAC6 (0.64) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28248162 0.77 HDAC6 (0.60) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL28865489 0.76 HDAC3 (0.55) HDAC6HDAC3HDAC1HDAC2GPR39

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699048-A Oxadiazolamide derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same 株式会社钟根堂 2018-10-23 CN disclosed