SCHEMBL28867159

SCHEMBL28867159

N#Cc1ncccc1-n1ccnn1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 11/20 0.40
CYP11B1 P15538 1/20 0.40
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
GRM1 Q13255 2/20 0.36
KEAP1 Q14145 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CHRNB2 P17787 1/20 0.35
CYP2B6 P20813 1/20 0.35
MAOA P21397 1/20 0.35
CYP2C19 P33261 1/20 0.35
CHRNA4 P43681 1/20 0.35
HTR3A P46098 1/20 0.35
CYP19A1 P11511 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5854751 0.79 ALDH1A1 (0.49) NOTUMCYP11B1HCRTR1HCRTR2GRM1
SCHEMBL21486439 0.78 NPC1 (0.45) NOTUMCYP11B1HCRTR1HCRTR2GRM1
SCHEMBL30633068 0.76 NOTUM (0.42) NOTUMHCRTR1HCRTR2KEAP1CYP1A2
SCHEMBL1587098 0.76 NOTUM (0.42) NOTUMHCRTR1HCRTR2KEAP1CYP1A2
SCHEMBL30664780 0.75 ALDH1A1 (0.52) CYP11B1GRM1CYP3A4CYP2D6CYP1A2
SCHEMBL12476256 0.74 NOTUM (0.41) NOTUMHCRTR1HCRTR2CYP1A2CYP2C9
SCHEMBL16113420 0.74 NOTUM (0.47) NOTUMHCRTR1HCRTR2KEAP1CYP1A2
SCHEMBL18284817 0.74 NOTUM (0.43) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL15552503 0.73 KDM4E (0.42) NOTUMCYP19A1
SCHEMBL16031459 0.73 NOTUM (0.40) NOTUMHCRTR1HCRTR2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105308048-B Substituted 2-azabicyclic compounds and their use as orexin receptor modulators 詹森药业有限公司 2019-10-08 CN disclosed
CN-108864093-A Substituted 2- Azabicyclic compound and their purposes as orexin receptor regulator 詹森药业有限公司 2018-11-23 CN disclosed