SCHEMBL28868430

SCHEMBL28868430

[CH2]Cc1nn(-c2ccc(Br)cc2)c(=O)n1Cc1cccc(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 11/20 0.56
TP53 P04637 1/20 0.48
ADORA3 P0DMS8 2/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CA P42336 1/20 0.46
MAPT P10636 2/20 0.44
CMA1 P23946 1/20 0.44
THRB P10828 1/20 0.44
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19643674 0.89 ROCK2 (0.56) ROCK2TP53ADORA3PIK3R1PIK3CA
SCHEMBL19643570 0.89 ROCK2 (0.58) ROCK2TP53ADORA3PIK3R1PIK3CA
SCHEMBL19644071 0.88 ROCK2 (0.72) ROCK2TP53ADORA3PIK3R1PIK3CA
SCHEMBL19643781 0.86 ROCK2 (0.67) ROCK2TP53PIK3R1PIK3CAMAPT
SCHEMBL19644451 0.84 ROCK2 (0.51) ROCK2TP53ADORA3PIK3R1PIK3CA
SCHEMBL19643227 0.81 ROCK2 (0.50) ROCK2TP53PIK3R1PIK3CAMAPT
SCHEMBL19643602 0.77 ROCK2 (0.60) ROCK2TP53PIK3R1PIK3CAMAPT
SCHEMBL19643876 0.73 ROCK2 (0.84) ROCK2
SCHEMBL19643173 0.72 ROCK2 (1.00) ROCK2
SCHEMBL19643096 0.71 ROCK2 (1.00) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153663-A Triazolones and Tetrazolones as ROCK Inhibitors 百时美施贵宝公司 2019-01-04 CN disclosed