SCHEMBL28868517

SCHEMBL28868517

O=Cc1ccnc(Br)c1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 1/20 0.53
TRIM33 Q9UPN9 1/20 0.53
CCR1 P32246 1/20 0.45
CCR5 P51681 1/20 0.45
CCR8 P51685 1/20 0.45
ERN1 O75460 4/20 0.33
TDP1 Q9NUW8 2/20 0.33
KMT2A Q03164 3/20 0.32
LMNA P02545 2/20 0.32
MEN1 O00255 2/20 0.32
THRB P10828 1/20 0.32
BLM P54132 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
ALDH1A1 P00352 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
HSP90AA1 P07900 1/20 0.30
IDO1 P14902 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL748190 0.80 CCR1 (0.50) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL30529332 0.80 CCR1 (0.50) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL27887406 0.78 TRIM24 (0.57) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL31207190 0.77 CCR1 (0.47) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL24265348 0.77 CCR1 (0.47) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL29950826 0.75 CCR1 (0.45) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL29954640 0.75 CCR1 (0.45) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL2894661 0.75 CCR1 (0.45) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL19139612 0.75 CCR1 (0.45) TRIM24TRIM33CCR1CCR5CCR8
SCHEMBL17512179 0.75 TRIM24 (0.53) TRIM24TRIM33CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232109-A PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 广东东阳光药业有限公司 2022-10-25 CN disclosed