SCHEMBL28870516

SCHEMBL28870516

COc1cccc(NC(=O)c2cc(OC)c(OC)cc2Br)c1

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.71
NPC1 O15118 5/20 0.71
TP53 P04637 2/20 0.67
SMN1; SMN2 Q16637 2/20 0.67
POLB P06746 1/20 0.66
KMT2A Q03164 2/20 0.61
RXFP1 Q9HBX9 1/20 0.59
KCNK3 O14649 1/20 0.59
KCNK9 Q9NPC2 1/20 0.59
USP2 O75604 1/20 0.59
NLRP3 Q96P20 1/20 0.58
ALDH1A1 P00352 1/20 0.58
PKM P14618 1/20 0.58
KDM4E B2RXH2 1/20 0.57
GAA P10253 1/20 0.57
HPGD P15428 1/20 0.57
PDE10A Q9Y233 1/20 0.56
LRRK2 Q5S007 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ether SCHEMBL28282920 0.93 NPC1 (0.62) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL1499642 0.83 RAB9A (1.00) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL30758588 0.83 RAB9A (1.00) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL25378644 0.82 HTT (0.56) RAB9ANPC1SMN1; SMN2KMT2ARXFP1
SCHEMBL4254148 0.78 RAB9A (0.76) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL4248720 0.78 RXFP1 (0.76) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL12468557 0.77 AVPR2 (0.75) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL18845166 0.77 KMT2A (0.82) RAB9ANPC1TP53SMN1; SMN2POLB
SCHEMBL10055020 0.76 NPC1 (0.94) RAB9ANPC1TP53SMN1; SMN2KMT2A
SCHEMBL4436642 0.76 KCNK3 (0.77) RAB9ANPC1TP53SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109369526-A A kind of synthetic method and its antitumor application thereof of nitidine derivative 桂林理工大学 2019-02-22 CN claimed
CN-109369526-A A kind of synthetic method and its antitumor application thereof of nitidine derivative 桂林理工大学 2019-02-22 CN disclosed