SCHEMBL28873228

SCHEMBL28873228

C[CH]Nc1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
GAA P10253 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
TGM2 P21980 2/20 0.39
RAPGEF4 Q8WZA2 1/20 0.39
F13A1 P00488 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL515529 0.74 ALDH1A1 (0.56) CYP2A6RAB9ANPC1CYP2D6CYP2C9
SCHEMBL4525438 0.74 TSHR (0.43) CYP2A6RAB9ANPC1GAASMN1; SMN2
SCHEMBL3083947 0.74 CA1 (0.43) CYP2A6RAB9ANPC1CYP2D6CYP2C9
SCHEMBL360732 0.72
SCHEMBL3893966 0.72 CYP2D6 (0.44) CYP2A6RAB9ANPC1CYP2D6CYP2C9
SCHEMBL5541980 0.70 CYP2D6 (0.47) CYP2A6RAB9ANPC1CYP2D6CYP2C9
SCHEMBL5541983 0.70 CYP2D6 (0.47) CYP2A6RAB9ANPC1CYP2D6CYP2C9
SCHEMBL467157 0.69
SCHEMBL10368399 0.69
SCHEMBL20335404 0.69 MEN1 (0.50) CYP2A6RAB9ANPC1GAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689639-A Spirolactams as ROCK inhibitor 百时美施贵宝公司 2019-04-26 CN disclosed