SCHEMBL28874489

SCHEMBL28874489

COc1ccc2oc(SCc3ccc(C(F)(F)F)cc3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.54
MAPT P10636 4/20 0.54
LMNA P02545 4/20 0.54
ALDH1A1 P00352 2/20 0.54
HTT P42858 2/20 0.54
NPSR1 Q6W5P4 1/20 0.49
GAA P10253 1/20 0.46
TSHR P16473 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
POLB P06746 1/20 0.46
NPC1 O15118 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2E1 P05181 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C8 P10632 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29878256 1.00 SMN1; SMN2 (0.54) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL28874291 0.85 GSK3B (0.48) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL28874494 0.85 ELANE (0.51) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL29878659 0.85 ELANE (0.51) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL22524936 0.84 ELANE (0.54) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL29032759 0.84 MAPT (0.64) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL29878407 0.83 LMNA (0.55) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL28874375 0.83 LMNA (0.55) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL22525010 0.82 ELANE (0.57) SMN1; SMN2MAPTLMNAALDH1A1HTT
SCHEMBL28874416 0.82 LMNA (0.46) SMN1; SMN2MAPTLMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124485-B Sulfoxide-containing benzoxazole derivative, and preparation method and application thereof 中国医学科学院药物研究所 2023-12-15 CN disclosed
CN-115124485-A Benzoxazole derivatives containing sulfoxide as well as preparation method and application thereof 中国医学科学院药物研究所 2022-09-30 CN disclosed