SCHEMBL28877840

SCHEMBL28877840

Nc1nc(N)c([N+](=O)[O-])c(-c2ccc(OC(F)F)cc2)n1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 1/20 0.44
ADORA1 P30542 3/20 0.41
ADORA2A P29274 1/20 0.41
MGMT P16455 8/20 0.41
DRD1 P21728 1/20 0.37
ROCK1 Q13464 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
DHFR P00374 2/20 0.35
EIF4E P06730 1/20 0.35
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
GRM2 Q14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29973964 1.00 MAPT (0.44) MAPTRAB9AMEN1NPC1KMT2A
SCHEMBL29974131 0.83 MGMT (0.40) MAPTRAB9AMEN1NPC1KMT2A
SCHEMBL28877904 0.83 MGMT (0.40) MAPTRAB9AMEN1NPC1KMT2A
SCHEMBL28957972 0.79 ADORA2A (0.47) MAPTRAB9AMEN1KMT2AADORA1
SCHEMBL29974285 0.73 HRH2 (0.42) MEN1KMT2AMGMTDHFRCCNA2
SCHEMBL12991933 0.69 MAPT (0.58) MAPTRAB9AMEN1NPC1KMT2A
SCHEMBL17667876 0.68 ADORA2A (0.54) MAPTRAB9AMEN1KMT2AADORA1
SCHEMBL27612801 0.68 PIK3CG (0.53) MAPTRAB9AMEN1KMT2AADORA1
SCHEMBL27612725 0.68 CD274 (0.46) MAPTRAB9ANPC1ADORA1ADORA2A
SCHEMBL9640554 0.67 MGMT (0.49) MAPTRAB9ANPC1KMT2AMGMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115141202-A Pyrimidopyrazinone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-04 CN disclosed