SCHEMBL28878366

SCHEMBL28878366

CC(C)(C)OC(=O)N(OC(=O)Nc1cc(F)ccc1Cl)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 3/20 0.40
PDK2 Q15119 3/20 0.40
PDK3 Q15120 3/20 0.40
PDK4 Q16654 3/20 0.40
KCNQ4 P56696 3/20 0.38
KCNQ5 Q9NR82 3/20 0.38
ALDH1A1 P00352 4/20 0.38
CLCN2 P51788 1/20 0.38
PYGL P06737 2/20 0.37
RAB9A P51151 1/20 0.36
NPC1 O15118 1/20 0.36
ALOX12 P18054 1/20 0.36
ALOX15 P16050 2/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4367386 0.79 CLCN2 (0.36) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL6856839 0.72 PDK1 (0.58) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL15614546 0.72 MAPT (0.51) KCNQ4KCNQ5ALDH1A1KMT2AMEN1
SCHEMBL28738831 0.72 PDK1 (0.56) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL292274 0.72 AAK1 (0.39) KCNQ4KCNQ5ALDH1A1CLCN2
SCHEMBL30227411 0.71 GRIK1 (0.48) KCNQ4KCNQ5CLCN2PYGLNPC1
SCHEMBL14085553 0.71 NPC1 (0.58) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL30227212 0.71 GRIK1 (0.48) KCNQ4KCNQ5CLCN2PYGLNPC1
SCHEMBL27398698 0.71 MAPT (0.51) KCNQ4KCNQ5ALDH1A1KMT2AMEN1
SCHEMBL3789950 0.71 CA12 (0.48) PDK1PDK2PDK3PDK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110325184-A Amide derivatives 第一三共株式会社 2019-10-11 CN disclosed