SCHEMBL28888596

SCHEMBL28888596

CCOC(C)n1cc(-c2ncnc3c2ccn3OC(=O)C(C)(C)CC)cn1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 7/20 0.37
JAK1 P23458 5/20 0.37
TYK2 P29597 3/20 0.37
JAK3 P52333 3/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
SIGMAR1 Q99720 1/20 0.34
MAP3K5 Q99683 2/20 0.32
CYP3A4 P08684 1/20 0.31
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31291526 0.84 JAK2 (0.37) JAK2JAK1TYK2JAK3HDAC3
SCHEMBL28857054 0.81 JAK2 (0.37) JAK2JAK1TYK2JAK3HDAC3
SCHEMBL30749812 0.80 JAK2 (0.37) JAK2JAK1TYK2JAK3HDAC3
SCHEMBL2605520 0.80 JAK2 (0.37) JAK2JAK1TYK2JAK3HDAC3
SCHEMBL17967357 0.79 SIGMAR1 (0.38) JAK2JAK1SIGMAR1CYP3A4
SCHEMBL28801738 0.79 JAK2 (0.56) JAK2JAK1TYK2JAK3HDAC6
SCHEMBL28801746 0.79 JAK2 (0.56) JAK2JAK1TYK2JAK3HDAC6
SCHEMBL26541045 0.78 JAK2 (0.42) JAK2JAK1TYK2JAK3HDAC3
SCHEMBL10247499 0.77 JAK2 (0.38) JAK2JAK1TYK2JAK3HDAC3
SCHEMBL28325796 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181103-A Preparation method of barretinib 上海博悦生物科技有限公司 2022-10-14 CN disclosed