SCHEMBL28889374

SCHEMBL28889374

Cc1ncccc1C(C(=O)NC(=S)NCC(F)F)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.39
GPR52 Q9Y2T5 1/20 0.35
ALDH1A1 P00352 4/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PHGDH O43175 2/20 0.33
TACR1 P25103 1/20 0.33
GAA P10253 1/20 0.33
KCNN4 O15554 1/20 0.33
DDR1 Q08345 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
NPSR1 Q6W5P4 3/20 0.32
POLB P06746 2/20 0.32
P2RX7 Q99572 1/20 0.32
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.32
ALOX12 P18054 1/20 0.32
KMT2A Q03164 1/20 0.32
SORT1 Q99523 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29893596 1.00 ADRB2 (0.39) ADRB2GPR52ALDH1A1L3MBTL1HTT
SCHEMBL28889291 0.92 ADRB2 (0.39) ADRB2ALDH1A1L3MBTL1HTTTDP1
SCHEMBL29893566 0.92 ADRB2 (0.39) ADRB2ALDH1A1L3MBTL1HTTTDP1
SCHEMBL29942367 0.91 ADRB2 (0.40) ADRB2GPR52ALDH1A1L3MBTL1TACR1
SCHEMBL28889279 0.90 ADRB2 (0.40) ADRB2GPR52ALDH1A1L3MBTL1HTT
SCHEMBL29942209 0.88 ADRB2 (0.38) ADRB2ALDH1A1L3MBTL1PHGDHGAA
SCHEMBL28889299 0.87 HDAC4 (0.40) ADRB2GPR52ALDH1A1HTTTDP1
SCHEMBL28889382 0.81 ADRB2 (0.39) ADRB2ALDH1A1L3MBTL1GAAKCNN4
SCHEMBL29942075 0.81 ADRB2 (0.42) ADRB2GPR52ALDH1A1L3MBTL1HTT
SCHEMBL29893632 0.80 ADRB2 (0.37) ADRB2ALDH1A1L3MBTL1HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed