SCHEMBL28890847

SCHEMBL28890847

O=C1Nc2ccccc2C1=Cc1ccc(-c2cn(-c3ccccc3Cl)nn2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.74
BCHE P06276 1/20 0.53
PDGFRB P09619 4/20 0.48
MEN1 O00255 2/20 0.48
ALDH1A1 P00352 2/20 0.48
APP P05067 2/20 0.48
MAPT P10636 2/20 0.48
MAPK1 P28482 2/20 0.48
SNCA P37840 2/20 0.48
KMT2A Q03164 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
CTRC Q99895 2/20 0.48
NPC1 O15118 1/20 0.48
GMNN O75496 1/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
MTOR P42345 1/20 0.48
RAB9A P51151 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28890846 1.00 KDR (0.74) KDRBCHEPDGFRBMEN1ALDH1A1
SCHEMBL29657663 0.89 KDR (0.80) KDRBCHEMEN1KMT2AFLT3
SCHEMBL28414342 0.89 KDR (0.80) KDRBCHEMEN1KMT2AFLT3
SCHEMBL28414341 0.89 KDR (0.80) KDRBCHEMEN1KMT2AFLT3
SCHEMBL28416374 0.88 KDR (0.79) KDRPDGFRBMEN1ALDH1A1APP
SCHEMBL28411671 0.88 KDR (0.74) KDRPDGFRBMEN1ALDH1A1APP
SCHEMBL28416371 0.88 KDR (0.79) KDRPDGFRBMEN1ALDH1A1APP
SCHEMBL28411669 0.88 KDR (0.74) KDRPDGFRBMEN1ALDH1A1APP
SCHEMBL28413621 0.86 KDR (0.84) KDRPDGFRBCTRCEGFRERBB2
SCHEMBL28410371 0.85 KDR (1.00) KDRPDGFRBERBB2RETFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153889-B 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2022-05-20 CN disclosed
CN-111153889-A 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2020-05-15 CN disclosed