SCHEMBL29657663

SCHEMBL29657663

O=C1Nc2ccc(F)cc2/C1=C/c1ccc(-c2cn(-c3ccccc3Cl)nn2)cc1

nearest known ligand 0.80

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.80
BCHE P06276 1/20 0.47
RPS6KA3 P51812 1/20 0.45
LRRK2 Q5S007 1/20 0.44
FLT3 P36888 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
RAF1 P04049 1/20 0.43
MDM2 Q00987 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28414341 1.00 KDR (0.80) KDRBCHERPS6KA3LRRK2FLT3
SCHEMBL28414342 1.00 KDR (0.80) KDRBCHERPS6KA3LRRK2FLT3
SCHEMBL29657615 0.91 KDR (0.83) KDRRPS6KA3LRRK2FLT3MEN1
SCHEMBL28415507 0.91 KDR (0.83) KDRRPS6KA3LRRK2FLT3MEN1
SCHEMBL28415508 0.91 KDR (0.83) KDRRPS6KA3LRRK2FLT3MEN1
SCHEMBL28414126 0.89 KDR (1.00) KDRRPS6KA3FLT3MEN1KMT2A
SCHEMBL29657627 0.89 KDR (1.00) KDRRPS6KA3FLT3MEN1KMT2A
SCHEMBL28414128 0.89 KDR (1.00) KDRRPS6KA3FLT3MEN1KMT2A
SCHEMBL28890846 0.89 KDR (0.74) KDRBCHEFLT3MEN1KMT2A
SCHEMBL28890847 0.89 KDR (0.74) KDRBCHEFLT3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153889-B 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2022-05-20 CN disclosed