SCHEMBL28895109

SCHEMBL28895109

N#CC1(Nc2cnc3c(c2)COC3=O)CCCC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
AR P10275 2/20 0.39
GAA P10253 2/20 0.36
PDE4A P27815 10/20 0.34
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
PDE7A Q13946 2/20 0.31
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28895292 0.77 CYP1A2 (0.50) CYP1A2GAAALDH1A1POLBJAK2
SCHEMBL28895242 0.76 CYP1A2 (0.49) CYP1A2GAAALDH1A1POLBJAK2
SCHEMBL28895284 0.75 CYP1A2 (0.41) CYP1A2GAAPDE4AALDH1A1POLB
SCHEMBL29580770 0.75 CYP1A2 (0.41) CYP1A2GAAPDE4AALDH1A1POLB
SCHEMBL28895136 0.74 CYP1A2 (0.47) CYP1A2GAAALDH1A1POLBJAK2
SCHEMBL29581246 0.72 AR (0.36) ARALDH1A1
SCHEMBL28895119 0.72 AR (0.36) ARALDH1A1
SCHEMBL25218349 0.64 MAOA (0.38) ARGAAJAK2
SCHEMBL29915220 0.64 MAOA (0.38) ARGAAJAK2
SCHEMBL28895140 0.64 MAPT (0.49) CYP1A2ARGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed