SCHEMBL28895238

SCHEMBL28895238

Cc1ncc(-c2ccc3cnc(NC(=O)CC4OCCNC4C)cc3c2)n1C

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 20/20 0.60
GSK3B P49841 18/20 0.60
WNT1 P04628 8/20 0.60
CLK2 P49760 2/20 0.56
CLK3 P49761 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28895293 0.87 GSK3B (0.62) DYRK1AGSK3BWNT1
SCHEMBL28895356 0.85 WNT1 (0.72) DYRK1AGSK3BWNT1
SCHEMBL19515496 0.84 DYRK1A (0.74) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL28895159 0.83 GSK3B (0.62) DYRK1AGSK3BWNT1
SCHEMBL28895330 0.83 GSK3B (0.61) DYRK1AGSK3BWNT1
SCHEMBL28895289 0.83 GSK3B (0.59) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL28895311 0.83 GSK3B (0.52) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL19515975 0.80 DYRK1A (0.73) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL19516077 0.78 GSK3B (0.73) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL19516080 0.78 GSK3B (0.73) DYRK1AGSK3BWNT1CLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311819-B Isoquinolin-3-yl carboxamides, their preparation and their use 萨穆梅德有限公司 2022-10-25 CN claimed