SCHEMBL28895256

SCHEMBL28895256

CCNc1cc(-c2ccc(Cl)cc2)nc(-c2cccnc2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.57
CYP2C9 P11712 3/20 0.57
DYRK1A Q13627 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
ADORA3 P0DMS8 3/20 0.49
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ROS1 P08922 1/20 0.46
KMT2A Q03164 3/20 0.46
PPARG P37231 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NR2E3 Q9Y5X4 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
PDE5A O76074 2/20 0.45
RXFP1 Q9HBX9 1/20 0.43
MEN1 O00255 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30085796 1.00 CYP3A4 (0.57) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL28895149 0.90 CYP3A4 (0.55) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL30085872 0.90 CYP3A4 (0.55) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL28894659 0.88 CYP3A4 (0.53) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL30085446 0.88 CYP3A4 (0.53) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL30085785 0.85 ALDH1A1 (0.62) CYP3A4CYP2C9DYRK1ACLK4ALDH1A1
SCHEMBL28894899 0.85 DYRK1A (0.53) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL30085787 0.85 DYRK1A (0.53) CYP3A4CYP2C9DYRK1ACLK4ADORA3
SCHEMBL28959741 0.85 ALDH1A1 (0.62) CYP3A4CYP2C9DYRK1ACLK4ALDH1A1
SCHEMBL28894909 0.85 CYP3A4 (0.50) CYP3A4CYP2C9DYRK1ACLK4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed