SCHEMBL28895299

SCHEMBL28895299

Cc1cc(NC(=O)OC(C)(C)C)cc(F)c1C=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA9 Q16790 1/20 0.44
RORC P51449 11/20 0.38
CYP17A1 P05093 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SYK P43405 1/20 0.36
EGLN2 Q96KS0 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18106503 0.91 CA12 (0.42) CA12CA1CA9RORCCYP17A1
SCHEMBL28895142 0.88 CA12 (0.41) CA12CA1CA9RORCCYP17A1
SCHEMBL16236847 0.82 CA12 (0.48) CA12CA1CA9RORCCYP17A1
SCHEMBL28895300 0.80 CA12 (0.43) CA12CA1CA9RORCCYP17A1
SCHEMBL28895283 0.79 CA12 (0.42) CA12CA1CA9RORCCYP17A1
SCHEMBL15076456 0.79 CA12 (0.42) CA12CA1CA9RORCCYP17A1
SCHEMBL16302366 0.78 CA12 (0.51) CA12CA1CA9CYP17A1EGLN2
SCHEMBL28895279 0.78 CA12 (0.41) CA12CA1CA9RORCCYP17A1
SCHEMBL12225074 0.77 CA12 (0.54) CA12CA1CA9CYP17A1SYK
SCHEMBL29178873 0.76 EGLN2 (0.42) CA12CA1CA9RORCCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed