SCHEMBL28895283

SCHEMBL28895283

Cc1cc(NC(=O)OC(C)(C)C)cc(F)c1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SYK P43405 1/20 0.37
RORC P51449 5/20 0.37
RARA P10276 2/20 0.37
RARG P13631 2/20 0.37
RARB P10826 1/20 0.37
EGLN2 Q96KS0 2/20 0.37
CYP17A1 P05093 2/20 0.36
PPARG P37231 1/20 0.35
LCK P06239 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17629762 0.91 RARA (0.43) CA12CA1CA9SYKRORC
SCHEMBL28895279 0.87 CA12 (0.41) CA12CA1CA9SYKRORC
SCHEMBL9288893 0.84 CYP3A4 (0.47) CA12CA1CA9MEN1KMT2A
SCHEMBL16236847 0.84 CA12 (0.48) CA12CA1CA9SYKRORC
SCHEMBL3120908 0.82 CA12 (0.48) CA12CA1CA9EGLN2CYP17A1
SCHEMBL28895300 0.81 CA12 (0.43) CA12CA1CA9SYKRORC
SCHEMBL17643122 0.81 CA12 (0.39) CA12CA1CA9SYKRORC
SCHEMBL16137967 0.81 MAPT (0.41) CA12CA1CA9SYKEGLN2
SCHEMBL16302366 0.80 CA12 (0.51) CA12CA1CA9MEN1KMT2A
SCHEMBL28895299 0.79 CA12 (0.44) CA12CA1CA9SYKRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed