SCHEMBL28895323

SCHEMBL28895323

CC(C)(C#N)Nc1ccc2c(c1)COC2=O

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
MAPT P10636 3/20 0.49
KDM4E B2RXH2 2/20 0.49
HSD17B10 Q99714 1/20 0.48
NR3C1 P04150 5/20 0.46
PGR P06401 5/20 0.46
NR3C2 P08235 3/20 0.46
IMPDH2 P12268 1/20 0.46
LMNA P02545 2/20 0.45
GAA P10253 1/20 0.45
PRF1 P14222 4/20 0.45
PKM P14618 2/20 0.44
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29580859 1.00 ALDH1A1 (0.51) ALDH1A1MAPTKDM4EHSD17B10NR3C1
SCHEMBL28895199 0.76 KDM4E (0.33) ALDH1A1MAPTKDM4EHSD17B10GAA
SCHEMBL29581246 0.76 AR (0.36) ALDH1A1
SCHEMBL29581802 0.76 KDM4E (0.33) ALDH1A1MAPTKDM4EHSD17B10GAA
SCHEMBL28895119 0.76 AR (0.36) ALDH1A1
SCHEMBL15727795 0.75 MKNK1 (0.46)
SCHEMBL15727792 0.73 PARP10 (0.51)
SCHEMBL5558567 0.72 MAPT (0.61) ALDH1A1MAPTKDM4EHSD17B10LMNA
SCHEMBL3624124 0.72 MAPT (0.55) ALDH1A1MAPTKDM4EHSD17B10NR3C1
SCHEMBL14177746 0.71 ALDH1A1 (0.44) ALDH1A1MAPTKDM4ENR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed