SCHEMBL28895600

SCHEMBL28895600

Nc1nc2c(s1)C(=O)C(N)CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
MAPK1 P28482 2/20 0.51
MAPT P10636 2/20 0.38
DRD3 P35462 5/20 0.37
DRD2 P14416 4/20 0.37
ATAD2 Q6PL18 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
HRH2 P25021 2/20 0.34
ADRA2A P08913 2/20 0.34
DRD4 P21917 2/20 0.34
ADRB2 P07550 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2B P18089 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597273 0.81 ALDH1A1 (0.50) ALDH1A1MAPK1MAPTDRD3DRD2
Bromide SCHEMBL6117488 0.79 ALDH1A1 (0.49) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL3802844 0.75 ALDH1A1 (0.56) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL13125933 0.73 ALDH1A1 (0.54) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL31572310 0.71 DRD3 (0.53) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL30784645 0.71 DRD3 (0.53) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL13125914 0.71 ALDH1A1 (0.78) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL13884489 0.70 ALDH1A1 (0.50) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL16879855 0.70 ALDH1A1 (0.40) ALDH1A1MAPK1MAPTDRD3DRD2
SCHEMBL13125920 0.69 ALDH1A1 (0.45) ALDH1A1MAPK1MAPTDRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111298127-A Composition comprising histamine release-promoting substance and inhibitory compound, and oral solid preparation containing the same 黄泳华 2020-06-19 CN disclosed