SCHEMBL28896283

SCHEMBL28896283

CC(C)(C)OC(=O)c1cncnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.46
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GPR119 Q8TDV5 1/20 0.36
GABRA1 P14867 4/20 0.36
GABRG2 P18507 4/20 0.36
GABRB3 P28472 4/20 0.36
GABRA3 P34903 4/20 0.36
GABRA2 P47869 4/20 0.36
ALDH1A1 P00352 3/20 0.36
ATM Q13315 1/20 0.36
SLC7A5 Q01650 1/20 0.36
HPGDS O60760 1/20 0.35
ELANE P08246 1/20 0.35
THRB P10828 1/20 0.35
GABRA5 P31644 3/20 0.35
GABRA4 P48169 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638364 0.81 CA1 (0.44) HCAR2CA12CA1CA2CA9
SCHEMBL2561603 0.79 HCAR2 (0.46) HCAR2ATM
SCHEMBL4872303 0.78 ABCG2 (0.50) CA12CA1CA2CA9CA14
SCHEMBL25659553 0.78 CA12 (0.40) CA12CA1CA2CA9CA14
SCHEMBL6258045 0.77 CYP2C19 (0.60) HCAR2CA12CA1CA2CA9
SCHEMBL29521617 0.77 CYP2C19 (0.60) HCAR2CA12CA1CA2CA9
SCHEMBL29350345 0.77 ALDH1A1 (0.66) HCAR2ALDH1A1ATMTHRBMAPT
SCHEMBL3654895 0.77 ALDH1A1 (0.66) HCAR2ALDH1A1ATMTHRBMAPT
SCHEMBL5366124 0.77 ATM (0.43) HCAR2CA12CA1CA2CA9
SCHEMBL1501699 0.77 ATM (0.40) HCAR2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111511744-B Diazaindole compounds 百时美施贵宝公司 2023-09-22 CN disclosed
CN-112823005-A Pyrrolopyrimidine ITK inhibitors 阿克拉瑞斯治疗股份有限公司 2021-05-18 CN disclosed
CN-111511744-A Diazaindole compounds 百时美施贵宝公司 2020-08-07 CN disclosed