SCHEMBL28898138

SCHEMBL28898138

Cc1c(C(=O)Nc2ccc(F)c(C#N)c2)c(F)c(C(=O)C(=O)NC(CF)C(F)F)n1C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.39
SLC10A1 Q14973 9/20 0.39
LRRK2 Q5S007 1/20 0.36
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
USP2 O75604 1/20 0.33
PGR P06401 1/20 0.33
AR P10275 1/20 0.32
BLM P54132 1/20 0.32
WRN Q14191 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28898134 0.93 SLC10A1 (0.42) GRM4SLC10A1LRRK2TSHRALDH1A1
SCHEMBL28898136 0.88 SLC10A1 (0.42) GRM4SLC10A1LRRK2
SCHEMBL28898130 0.86 SLC10A1 (0.41) GRM4SLC10A1LRRK2
SCHEMBL21408395 0.84 SLC10A1 (0.46) GRM4SLC10A1LRRK2ALDH1A1KDM4E
SCHEMBL21408396 0.84 SLC10A1 (0.46) GRM4SLC10A1LRRK2ALDH1A1KDM4E
SCHEMBL21428333 0.84 GRM4 (0.43) GRM4SLC10A1LRRK2TSHRALDH1A1
SCHEMBL28898148 0.83 GRM4 (0.39) GRM4SLC10A1LRRK2ALDH1A1KDM4E
SCHEMBL21408335 0.82 GRM4 (0.47) GRM4SLC10A1LRRK2TSHRALDH1A1
SCHEMBL28898147 0.82 TSHR (0.43) SLC10A1TSHRALDH1A1POLBMAPT
SCHEMBL28898160 0.81 TSHR (0.42) SLC10A1TSHRALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868026-B Capsid protein assembly inhibitor containing N-heterocyclic five-membered ring, pharmaceutical composition and application thereof 正大天晴药业集团股份有限公司 2022-11-25 CN disclosed