SCHEMBL28898147

SCHEMBL28898147

Cc1c(C(=O)Nc2ccc(F)c(F)c2)c(C)n(C)c1C(=O)C(=O)NC(CF)C(F)F

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 2/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SLC10A1 Q14973 13/20 0.39
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28898160 0.93 TSHR (0.42) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL28898154 0.92 SLC10A1 (0.46) TSHRSMN1; SMN2SLC10A1NPC1RAB9A
SCHEMBL28898135 0.92 TSHR (0.41) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL28898224 0.90 TSHR (0.46) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL28898134 0.89 SLC10A1 (0.42) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL28898150 0.89 TSHR (0.42) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL28898131 0.88 MAPT (0.42) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL21427912 0.86 TSHR (0.44) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL21810153 0.84 MAPT (0.51) TSHRMAPTSMN1; SMN2LMNAUSP2
SCHEMBL30095297 0.84 MAPT (0.51) TSHRMAPTSMN1; SMN2LMNAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868026-B Capsid protein assembly inhibitor containing N-heterocyclic five-membered ring, pharmaceutical composition and application thereof 正大天晴药业集团股份有限公司 2022-11-25 CN disclosed