SCHEMBL28898152

SCHEMBL28898152

Cn1c(C(=O)C(=O)NC(CF)C(F)F)cc(C(=O)Nc2ccc(F)c(C#N)c2)c1F

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.40
FSCN1 Q16658 1/20 0.35
SLC10A1 Q14973 8/20 0.35
RAB9A P51151 2/20 0.33
PGR P06401 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KCNH2 Q12809 1/20 0.33
AR P10275 1/20 0.33
BLM P54132 1/20 0.33
WRN Q14191 1/20 0.33
AKT1 P31749 1/20 0.32
LRRK2 Q5S007 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28898141 0.84 GRM4 (0.40) GRM4FSCN1SLC10A1RAB9APGR
SCHEMBL21427803 0.84 GRM4 (0.41) GRM4FSCN1SLC10A1RAB9ANPC1
SCHEMBL28902794 0.84 GRM4 (0.41) GRM4FSCN1SLC10A1RAB9ANPC1
SCHEMBL30294232 0.84 GRM4 (0.41) GRM4FSCN1SLC10A1RAB9ANPC1
SCHEMBL28898148 0.82 GRM4 (0.39) GRM4FSCN1SLC10A1PGRALDH1A1
SCHEMBL28898136 0.82 SLC10A1 (0.42) GRM4SLC10A1LRRK2
SCHEMBL30094001 0.81 GRM4 (0.44) GRM4FSCN1SLC10A1RAB9ANPC1
SCHEMBL21427892 0.81 GRM4 (0.44) GRM4FSCN1SLC10A1RAB9ANPC1
SCHEMBL28898138 0.81 GRM4 (0.39) GRM4SLC10A1PGRPOLBMAPT
SCHEMBL28898134 0.81 SLC10A1 (0.42) GRM4SLC10A1MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868026-B Capsid protein assembly inhibitor containing N-heterocyclic five-membered ring, pharmaceutical composition and application thereof 正大天晴药业集团股份有限公司 2022-11-25 CN disclosed