SCHEMBL28898159

SCHEMBL28898159

CCOC(=O)c1cc(C(=O)C(=O)NC(CF)C(F)F)n(C)c1COC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.35
SMAD3 P84022 1/20 0.35
KDM4E B2RXH2 6/20 0.34
HSD17B10 Q99714 5/20 0.34
ALDH1A1 P00352 5/20 0.34
HPGD P15428 4/20 0.34
GAA P10253 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.32
KMT2A Q03164 4/20 0.32
TSHR P16473 2/20 0.32
MEN1 O00255 1/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA7 P43166 2/20 0.32
CA9 Q16790 2/20 0.32
CA14 Q9ULX7 2/20 0.32
BAZ2B Q9UIF8 1/20 0.31
BAZ2A Q9UIF9 1/20 0.31
LMNA P02545 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28898140 0.87
SCHEMBL25645243 0.85 ESR1 (0.39) ESR1SMAD3KDM4EHSD17B10ALDH1A1
SCHEMBL28987381 0.82 ESR1 (0.36) ESR1SMAD3KDM4EHSD17B10ALDH1A1
SCHEMBL21428059 0.82 ESR1 (0.36) ESR1SMAD3KDM4EHSD17B10ALDH1A1
SCHEMBL21408306 0.77 KDM4E (0.43) ESR1SMAD3KDM4EHSD17B10ALDH1A1
SCHEMBL25645241 0.70 MAPT (0.37) KDM4EHSD17B10ALDH1A1HPGDGAA
SCHEMBL28898157 0.70 CYP1A2 (0.36) KDM4ESMN1; SMN2MAPT
SCHEMBL28898144 0.69 KMT2A (0.41) KDM4EALDH1A1HPGDGAASMN1; SMN2
SCHEMBL22906212 0.68 PHGDH (0.30)
SCHEMBL28486708 0.68 PHGDH (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868026-B Capsid protein assembly inhibitor containing N-heterocyclic five-membered ring, pharmaceutical composition and application thereof 正大天晴药业集团股份有限公司 2022-11-25 CN disclosed