SCHEMBL28899166

SCHEMBL28899166

O=C=NCCc1cccc(Br)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.52
MIF P14174 3/20 0.44
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
PYCR1 P32322 1/20 0.41
MAOB P27338 1/20 0.40
GPR84 Q9NQS5 1/20 0.39
TRPA1 O75762 1/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
HIF1A Q16665 1/20 0.39
CYP2A13 Q16696 1/20 0.39
EPAS1 Q99814 1/20 0.39
CYP11B1 P15538 1/20 0.38
ADRA2C P18825 1/20 0.38
CYP11B2 P19099 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804290 0.87 MIF (0.50) TAAR1MIFMAOBTRPA1CYP2E1
SCHEMBL8486630 0.81 TAAR1 (0.46) TAAR1MIFIDO1AGXTPYCR1
SCHEMBL14015247 0.80 MIF (0.45) TAAR1MIFTRPA1CYP2E1CYP2A6
SCHEMBL29542006 0.80 HTR3E (0.54) TAAR1MIFIDO1AGXTPYCR1
SCHEMBL1851734 0.80 HTR3E (0.54) TAAR1MIFIDO1AGXTPYCR1
SCHEMBL30829275 0.79 TAAR1 (0.52) TAAR1MIFIDO1AGXT
SCHEMBL13139339 0.79 TAAR1 (0.52) TAAR1MIFIDO1AGXT
SCHEMBL9178534 0.77 MIF (0.42) TAAR1MIFTRPA1CYP2E1CYP2A6
SCHEMBL28173860 0.77 MIF (0.46) MIFAGXTGPR84TRPA1CYP2E1
SCHEMBL1844610 0.77 TAAR1 (0.45) TAAR1MIFIDO1PYCR1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed