SCHEMBL28899201

SCHEMBL28899201

O=C1NC2(CC2)c2ccc([N+](=O)[O-])cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
CAPN9 O14815 1/20 0.54
CASP3 P42574 1/20 0.54
TDP2 O95551 3/20 0.50
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PTPRC P08575 3/20 0.46
S100A4 P26447 2/20 0.46
EGFR P00533 1/20 0.45
CA9 Q16790 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
MAPT P10636 1/20 0.43
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
CES1 P23141 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30095520 1.00 CYP3A4 (0.54) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL2144836 0.81 TDP1 (0.57) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL11523350 0.77 TDP1 (0.53) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL22855674 0.76 CYP3A4 (0.51) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL1950552 0.76 TDP2 (0.58) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL17434341 0.75 CYP3A4 (0.54) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL445340 0.74 CYP3A4 (0.53) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL22855479 0.74 CYP3A4 (0.49) CYP3A4TDP1CAPN9CASP3TDP2
SCHEMBL16006554 0.73 PBRM1 (0.42) CYP3A4TDP2PTPRCEGFRCA9
SCHEMBL22898415 0.73 CA9 (0.39) CYP3A4TDP1TDP2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed