SCHEMBL28905830

SCHEMBL28905830

Nc1nccc(-c2ccccc2OC(F)(F)F)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPL P40238 1/20 0.48
AURKA O14965 1/20 0.47
HSP90AA1 P07900 1/20 0.47
PRKACA P17612 1/20 0.47
ADORA2A P29274 1/20 0.47
CDK2 P24941 2/20 0.45
CCNT1 O60563 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK9 P50750 1/20 0.45
DYRK1A Q13627 4/20 0.44
GSK3B P49841 4/20 0.44
CDK5 Q00535 2/20 0.44
CDK5R1 Q15078 2/20 0.44
MAP3K14 Q99558 2/20 0.44
CLK1 P49759 1/20 0.44
FEN1 P39748 3/20 0.44
ALOX5AP P20292 1/20 0.44
HTR1A P08908 1/20 0.44
HTR7 P34969 1/20 0.44
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362587 0.80 HSP90AA1 (0.60) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL30507329 0.80 HSP90AA1 (0.60) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL30507526 0.79 HSP90AA1 (0.47) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL28512809 0.79 HSP90AA1 (0.47) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL3398117 0.78 MPL (0.44) MPLHSP90AA1ADORA2AFEN1ALOX5AP
SCHEMBL30507528 0.77 HSP90AA1 (0.53) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL30507237 0.77 CDK5 (0.58) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL28511492 0.77 CDK5 (0.58) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL28501185 0.77 HSP90AA1 (0.53) AURKAHSP90AA1PRKACAADORA2ACDK2
SCHEMBL935401 0.76 KMO (0.60) AURKAHSP90AA1PRKACAADORA2ACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-A Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2020-12-01 CN disclosed