SCHEMBL28906224

SCHEMBL28906224

C[Si](C)(C)CCOCn1nc(C#N)c2cc(Br)ccc21

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.41
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.30
PFKFB2 O60825 1/20 0.30
PFKFB1 P16118 1/20 0.30
PFKFB3 Q16875 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30138980 1.00 DGAT1 (0.41) DGAT1NPC1SMN1; SMN2GAANPSR1
SCHEMBL2471306 0.86 NPC1 (0.35) DGAT1NPC1PFKFB2PFKFB1PFKFB3
SCHEMBL31512383 0.83 ELANE (0.40) DGAT1NPC1SMN1; SMN2
SCHEMBL17849502 0.83 ELANE (0.40) DGAT1NPC1SMN1; SMN2
SCHEMBL4312796 0.83 DGAT1 (0.43) DGAT1NPC1
SCHEMBL3355074 0.81 DGAT1 (0.43) DGAT1NPC1
SCHEMBL2030421 0.81 DGAT1 (0.43) DGAT1NPC1
SCHEMBL20163415 0.81 DGAT1 (0.47) DGAT1NPC1SMN1; SMN2NPSR1
SCHEMBL14442048 0.81 ELANE (0.47) SMN1; SMN2GAA
SCHEMBL23042316 0.81 DGAT1 (0.44) DGAT1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117412967-A Methionine adenosine transferase 2A inhibitors 南京正大天晴制药有限公司 2024-01-16 CN disclosed
CN-115433211-A Pyrazidopyridone methionine adenosyltransferase 2A inhibitors 南京正大天晴制药有限公司 2022-12-06 CN disclosed