SCHEMBL28907192

SCHEMBL28907192

O=Cc1ccc(O[C@H]2CCOC2)nc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.43
ALDH1A1 P00352 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 2/20 0.41
EGFR P00533 2/20 0.39
ITK Q08881 2/20 0.39
LRRK2 Q5S007 2/20 0.36
NAMPT P43490 1/20 0.36
POLB P06746 1/20 0.36
GPR119 Q8TDV5 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
KRAS P01116 1/20 0.35
SOS1 Q07889 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL796051 1.00 ACACB (0.43) ACACBALDH1A1L3MBTL1KDM4EEGFR
SCHEMBL28530061 1.00 ACACB (0.43) ACACBALDH1A1L3MBTL1KDM4EEGFR
SCHEMBL30484274 0.91 ALDH1A1 (0.43) ACACBALDH1A1L3MBTL1KDM4ENAMPT
SCHEMBL26458925 0.91 ALDH1A1 (0.43) ACACBALDH1A1L3MBTL1KDM4ENAMPT
SCHEMBL28522216 0.88 ALDH1A1 (0.45) ACACBALDH1A1L3MBTL1KDM4EPOLB
SCHEMBL14480299 0.84 ACACB (0.42) ACACBEGFRITKNAMPTGPR119
SCHEMBL14480338 0.84 ACACB (0.42) ACACBEGFRITKNAMPTGPR119
SCHEMBL23147699 0.83 ALDH1A1 (0.49) ALDH1A1L3MBTL1KDM4ENAMPTPOLB
SCHEMBL30222191 0.83 ALDH1A1 (0.49) ALDH1A1L3MBTL1KDM4ENAMPTPOLB
SCHEMBL28520364 0.82 P4HTM (0.45) ACACBKDM4EEGFRITKNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409360-B Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2022-12-23 CN disclosed
CN-112409360-A Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2021-02-26 CN disclosed