SCHEMBL28907770

SCHEMBL28907770

CCOC(=O)c1conc1-c1cnc(C(F)(F)F)c(C)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.47
IDO1 P14902 1/20 0.44
NPSR1 Q6W5P4 1/20 0.39
HPGD P15428 3/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 5/20 0.38
JUN P05412 4/20 0.38
NFKB2 Q00653 4/20 0.38
RELA Q04206 4/20 0.38
MAPT P10636 5/20 0.37
ALDH1A1 P00352 5/20 0.36
GAA P10253 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GLA P06280 1/20 0.36
ATF1 P18846 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28527516 0.85 ALDH1A1 (0.39) KDM4EHPGDTSHRMAPTALDH1A1
SCHEMBL21590765 0.81 KDM4E (0.42) KDM4EIDO1HPGDCASP1CASP7
SCHEMBL28526135 0.79 TSHR (0.37) KDM4EHPGDCASP1CASP7HSD17B10
SCHEMBL262187 0.78 KDM4E (0.52) KDM4EIDO1NPSR1HPGDCASP1
SCHEMBL28521042 0.78 TSHR (0.36) KDM4EHPGDHSD17B10TSHRMAPT
SCHEMBL5773409 0.78 MAPT (0.49) KDM4EIDO1NPSR1TSHRNFKB1
SCHEMBL11396911 0.77 MEN1 (0.53) KDM4EHPGDCASP1CASP7HSD17B10
SCHEMBL20241126 0.77 ALDH1A1 (0.42) HSD17B10TSHRMAPTALDH1A1SMN1; SMN2
SCHEMBL3978092 0.75 JAK2 (0.55) KDM4ENPSR1HPGDHSD17B10TSHR
SCHEMBL18149813 0.74 KDM4E (0.58) KDM4EIDO1NPSR1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112424196-A Novel isoxazolyl ether derivatives as GABAA alpha 5 PAM 豪夫迈·罗氏有限公司 2021-02-26 CN disclosed