SCHEMBL28908138

SCHEMBL28908138

O=C(Nc1cnc2ccccc2c1)OBr

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.62
KDM4E B2RXH2 7/20 0.61
RAB9A P51151 10/20 0.59
NPC1 O15118 10/20 0.59
SMN1; SMN2 Q16637 7/20 0.59
MAPT P10636 2/20 0.59
NFKB1 P19838 1/20 0.59
NFKB2 Q00653 1/20 0.59
RELA Q04206 1/20 0.59
ALDH1A1 P00352 3/20 0.58
POLB P06746 2/20 0.58
NPSR1 Q6W5P4 1/20 0.57
HSD17B10 Q99714 4/20 0.57
LMNA P02545 2/20 0.57
TSHR P16473 2/20 0.57
MITF O75030 1/20 0.57
XBP1 P17861 1/20 0.57
PAX8 Q06710 1/20 0.57
KLF5 Q13887 1/20 0.57
NOTUM Q6P988 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568774 0.86 KDM4E (0.67) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL4108874 0.82 KDR (0.63) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL27866684 0.82 NPC1 (0.80) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL240482 0.81 TRPV1 (0.61) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL651159 0.81 KDR (0.74) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL879571 0.80 KDM4E (0.70) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL3994400 0.80 NPSR1 (0.71) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL14461305 0.80 HDAC1 (0.72) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL27617535 0.80 KDR (0.68) KDRKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL8397726 0.79 TRPV1 (0.58) KDRKDM4ERAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112375037-A Synthetic method of 3-amino-5-bromoquinoline 苏州康润医药有限公司 2021-02-19 CN claimed
CN-112375037-B Synthetic method of 3-amino-5-bromoquinoline 苏州康润医药有限公司 2022-04-12 CN disclosed
CN-112375037-A Synthetic method of 3-amino-5-bromoquinoline 苏州康润医药有限公司 2021-02-19 CN disclosed