SCHEMBL289157

SCHEMBL289157

CCCC(C(=O)O)c1ccc(C(=N)N)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPN1 P15169 1/20 0.67
CPB2 Q96IY4 1/20 0.67
F10 P00742 6/20 0.48
F2 P00734 6/20 0.48
PRSS1 P07477 5/20 0.46
PRSS2 P07478 3/20 0.46
PRSS3 P35030 3/20 0.46
F7 P08709 2/20 0.46
F3 P13726 2/20 0.46
TMPRSS15 P98073 1/20 0.44
PLG P00747 1/20 0.42
C1S P09871 1/20 0.42
LMNA P02545 1/20 0.42
NQO2 P16083 2/20 0.41
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
POLB P06746 2/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
TPSAB1 Q15661 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7370118 0.98 CPN1 (0.65) CPN1CPB2F10F2PRSS1
SCHEMBL9147869 0.82 F10 (0.53) CPN1CPB2F10F2PRSS1
SCHEMBL10957721 0.81 GRM8 (0.44) CPN1CPB2LMNACYP2C9CYP2C19
SCHEMBL4104203 0.80 HSD17B10 (0.43) CPN1CPB2F10PRSS1PRSS2
SCHEMBL22712583 0.80 LMNA (0.42) CPN1CPB2LMNACYP2C9CYP2C19
Hydrochloric Acid SCHEMBL11656002 0.79 CYP2C9 (0.46) CPN1CPB2LMNACYP2C9CYP2C19
SCHEMBL21295020 0.79 CPN1 (0.64) CPN1CPB2
SCHEMBL4100564 0.79 GAA (0.47) CPN1CPB2LMNACYP2C9CYP2C19
SCHEMBL633268 0.78 ESR1 (0.49) LMNACYP2C9CYP2C19GAA
SCHEMBL4269790 0.78 POLB (0.51) POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427476-A1 BETA-HAIRPIN PEPTIDOMIMETICS HAVING CXCR4 ANTAGONIZING ACTIVITY Polyphor Ag (CH) 2012-03-14 EP disclosed
WO-2010127704-A1 BETA-HAIRPIN PEPTIDOMIMETICS HAVING CXCR4 ANTAGONIZING ACTIVITY POLYPHOR AG (CH) 2010-11-11 WO disclosed
US-5441974-A Phenyl amidines lactones useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-08-15 US disclosed
WO-1993012103-A1 PHENYL AMIDINES LACTONES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-06-24 WO disclosed