Amitrole

Amitrole

SCHEMBL2892142

CC(=O)O.Nc1nc[nH]n1.O=CO

nearest known ligand 0.35

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Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Amitrole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MGMT P16455 2/20 0.35
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amitrole SCHEMBL2898789 0.92 MGMT (0.38) MGMTGAA
Amitrole SCHEMBL2892139 0.90
Amitrole SCHEMBL788110 0.77 HSP90AA1 (0.33)
Amitrole SCHEMBL44637 0.77
Trifluoroacetic Acid SCHEMBL508966 0.76 HRH4 (0.37)
Amitrole SCHEMBL31379743 0.75
Amitrole SCHEMBL10399233 0.75
Amitrole SCHEMBL11745846 0.74 KDM4E (0.32)
Amitrole SCHEMBL1172473 0.71 RXFP1 (0.45)
Amitrole SCHEMBL7401602 0.67 CDK1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2259665-A1 Solution for surface treatment MEC COMPANY LTD. (JP) 2010-12-08 EP disclosed