SCHEMBL28922237

SCHEMBL28922237

Cc1onc(-c2ccccc2)c1-c1ccc(S(=O)(=O)NS(=O)(=O)c2ccc(-c3c(-c4ccccc4)noc3C)cc2)cc1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.82
MT-CO2 P00403 3/20 0.82
PTGS1 P23219 5/20 0.73
CA12 O43570 1/20 0.73
CA1 P00915 1/20 0.73
CA2 P00918 1/20 0.73
LMNA P02545 1/20 0.73
CA3 P07451 1/20 0.73
ADRB2 P07550 1/20 0.73
ADRB1 P08588 1/20 0.73
CYP3A4 P08684 1/20 0.73
ADORA3 P0DMS8 1/20 0.73
CHRM1 P11229 1/20 0.73
ADRA2B P18089 1/20 0.73
CA4 P22748 1/20 0.73
CA6 P23280 1/20 0.73
SLC6A2 P23975 1/20 0.73
PDE4A P27815 1/20 0.73
ADORA1 P30542 1/20 0.73
CA5A P35218 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30958763 0.92 PTGS2 (0.75) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL5481289 0.90 PTGS2 (1.00) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL5071844 0.90 PTGS2 (0.81) PTGS2MT-CO2PTGS1CA12CA1
Water SCHEMBL5477391 0.89 PTGS2 (1.00) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL5073588 0.88 PTGS2 (0.81) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL5071050 0.88 PTGS2 (0.77) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL28961699 0.87 PTGS2 (0.79) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL5069852 0.87 PTGS2 (0.75) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL5586953 0.87 PTGS2 (0.75) PTGS2MT-CO2PTGS1CA12CA1
SCHEMBL11925221 0.87 PTGS2 (0.75) PTGS2MT-CO2PTGS1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111978266-B Parecoxib sodium, injection preparation and preparation method 四川制药制剂有限公司 2021-09-14 CN disclosed
CN-111978266-A Parecoxib sodium, injection preparation and preparation method 四川制药制剂有限公司 2020-11-24 CN disclosed