SCHEMBL289267

SCHEMBL289267

CN1Cc2cc(-c3ccc(C(N)C(C=O)NC(=O)C4(NC(=O)O)CCOCC4)cc3)ccc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSC P53634 10/20 0.43
CTSK P43235 6/20 0.43
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
SDCBP O00560 1/20 0.34
SDC2 P34741 1/20 0.34
UGCG Q16739 2/20 0.33
OPRD1 P41143 1/20 0.32
PRF1 P14222 1/20 0.31
CHRM4 P08173 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299705 0.80 CTSC (0.51) CTSCCTSKPIK3CAMTORSDCBP
SCHEMBL2890645 0.78 CTSC (0.68) CTSCCTSK
SCHEMBL289266 0.78 CTSC (0.47) CTSCCTSKPIK3CAMTORSDCBP
SCHEMBL290587 0.77 TACR2 (0.32)
SCHEMBL298896 0.74 CTSC (0.59) CTSCCTSKSDCBPSDC2
SCHEMBL2892971 0.70 CTSC (0.48) CTSCCTSKSDCBPSDC2UGCG
SCHEMBL2892969 0.70 CTSC (0.48) CTSCCTSKSDCBPSDC2UGCG
SCHEMBL2890558 0.68 CTSC (0.62) CTSCCTSK
SCHEMBL2890557 0.68 CTSC (0.62) CTSCCTSK
SCHEMBL299126 0.68 CTSC (0.43) CTSCCTSKSDCBPSDC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed