SCHEMBL28933265

SCHEMBL28933265

c1ccc2c(c1)ccn2-c1ccnc(NCCN2CCCC2)n1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 11/20 0.82
MKNK2 Q9HBH9 9/20 0.64
MAPK8 P45983 2/20 0.52
MAPK9 P45984 2/20 0.52
MAPK10 P53779 1/20 0.52
CDK2 P24941 2/20 0.49
CDC7 O00311 1/20 0.49
ROCK1 Q13464 1/20 0.49
JUN P05412 1/20 0.48
CXCR4 P61073 1/20 0.46
HRH3 Q9Y5N1 2/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
SLC6A2 P23975 1/20 0.44
HRH2 P25021 1/20 0.44
HTR1D P28221 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR7 P34969 1/20 0.44
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18803539 0.90 MKNK1 (1.00) MKNK1MKNK2MAPK8MAPK9MAPK10
SCHEMBL18803637 0.82 MKNK1 (0.70) MKNK1MKNK2MAPK8MAPK9MAPK10
SCHEMBL1089672 0.79 CXCR4 (0.72) MKNK1CXCR4HRH3ADRA2BADRA2C
SCHEMBL18803570 0.78 MKNK1 (1.00) MKNK1MKNK2CDK2CDC7ROCK1
SCHEMBL28690595 0.78 MKNK1 (0.52) MKNK1MKNK2MAPK8MAPK9MAPK10
SCHEMBL29353130 0.78 MKNK1 (0.52) MKNK1MKNK2MAPK8MAPK9MAPK10
SCHEMBL28704767 0.77 MKNK1 (0.64) MKNK1MKNK2MAPK8MAPK9MAPK10
SCHEMBL18803525 0.73 MKNK1 (1.00) MKNK1MKNK2LCK
SCHEMBL18803544 0.73 MKNK1 (1.00) MKNK1MKNK2MAPK8MAPK9MAPK10
SCHEMBL5094294 0.72 MAPK8 (0.78) MKNK1MKNK2MAPK8MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113956240-A Pyrimidine derivatives and application thereof in preparing antitumor drugs 陕西师范大学 2022-01-21 CN claimed
CN-113956240-B Pyrimidine derivatives and application thereof in preparing antitumor drugs 陕西师范大学 2023-02-14 CN disclosed
CN-113956240-A Pyrimidine derivatives and application thereof in preparing antitumor drugs 陕西师范大学 2022-01-21 CN disclosed