SCHEMBL28934239

SCHEMBL28934239

COc1cc(C)ccc1-c1nnc(Cl)c2cc(C(F)(F)F)ccc12

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.48
SCN9A Q15858 14/20 0.40
CRHR1 P34998 2/20 0.39
KIF11 P52732 2/20 0.39
SPR P35270 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28934436 0.87 ACHE (0.41) PDE5ASCN9ACRHR1
SCHEMBL28963081 0.86 SCN9A (0.40) PDE5ASCN9ACRHR1KIF11
SCHEMBL31309258 0.84 PDE5A (0.46) PDE5ASCN9ACRHR1SPR
SCHEMBL28934449 0.84 KDM4E (0.40) PDE5ASCN9ACRHR1KIF11
SCHEMBL28934496 0.84 PDE5A (0.46) PDE5ASCN9ACRHR1
SCHEMBL28934710 0.82 ACHE (0.41) PDE5ASCN9ACRHR1
SCHEMBL28934326 0.81 ACHE (0.36) PDE5ASCN9ACRHR1
SCHEMBL30108833 0.81 ACHE (0.36) PDE5ASCN9ACRHR1
SCHEMBL28934464 0.81 MAPT (0.40) CRHR1
SCHEMBL30181352 0.80 SCN9A (0.46) PDE5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed