SCHEMBL28934472

SCHEMBL28934472

COc1cc(C)ccc1-c1n[nH]c(=O)c2c(F)cccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
SCN9A Q15858 3/20 0.39
PDE7A Q13946 3/20 0.38
TNKS O95271 3/20 0.37
TNKS2 Q9H2K2 2/20 0.37
ROCK1 Q13464 1/20 0.36
PARP1 P09874 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
PRMT1 Q99873 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
AR P10275 2/20 0.34
MAPT P10636 2/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30101063 1.00 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL28934306 0.91 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL30101072 0.88 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL30108722 0.86 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL28934651 0.86 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL30101115 0.81 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL28934442 0.79 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL30108665 0.79 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DSCN9A
SCHEMBL28934465 0.76 MAPT (0.35) SCN9APDE7ACYP2C9CYP2C19MAPT
SCHEMBL28934538 0.74 SCN9A (0.48) PDE4APDE4BPDE4CPDE4DSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed