SCHEMBL28938677

SCHEMBL28938677

CCc1cnc(-c2cc(OC)c3ncnc(NCc4ccc(C)nn4)c3c2)s1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 3/20 0.44
P2RX2 Q9UBL9 3/20 0.44
PDE5A O76074 12/20 0.41
CLK4 Q9HAZ1 3/20 0.40
MAPK1 P28482 2/20 0.40
USP2 O75604 2/20 0.40
LMNA P02545 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29481207 1.00 P2RX3 (0.44) P2RX3P2RX2PDE5ACLK4MAPK1
SCHEMBL22714768 0.90 P2RX3 (0.45) P2RX3P2RX2PDE5ACLK4MAPK1
SCHEMBL29481339 0.90 P2RX3 (0.45) P2RX3P2RX2PDE5ACLK4MAPK1
SCHEMBL28726527 0.88 P2RX3 (0.45) P2RX3P2RX2PDE5ACLK4MAPK1
SCHEMBL29481254 0.88 P2RX3 (0.45) P2RX3P2RX2PDE5ACLK4MAPK1
SCHEMBL29481280 0.85 CLK4 (0.40) PDE5ACLK4MAPK1USP2LMNA
SCHEMBL22714717 0.85 CLK4 (0.40) PDE5ACLK4MAPK1USP2LMNA
SCHEMBL28726614 0.83 CLK4 (0.39) PDE5ACLK4MAPK1USP2LMNA
SCHEMBL29481335 0.83 CLK4 (0.39) PDE5ACLK4MAPK1USP2LMNA
SCHEMBL29481199 0.82 CLK4 (0.42) PDE5ACLK4MAPK1USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118239931-A As P2X3Aminoquinazoline derivatives of inhibitors 奇斯药制品公司 2024-06-25 CN claimed
CN-114269432-B As P2X3Aminoquinazoline derivatives of inhibitors 奇斯药制品公司 2024-05-07 CN claimed
CN-114269432-A As P2X3Aminoquinazoline derivatives as inhibitors 奇斯药制品公司 2022-04-01 CN claimed