SCHEMBL28939463

SCHEMBL28939463

CC(C)(C)OC(=O)N1CCN(c2ccc(C#N)c3ncncc23)CC1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 5/20 0.51
RPS6KB1 P23443 9/20 0.46
AKT1 P31749 2/20 0.45
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45
EGLN2 Q96KS0 1/20 0.44
RET P07949 2/20 0.43
MAP4K4 O95819 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30161982 0.83 RPS6KB1 (0.54) GPR119RPS6KB1AKT1MAP4K4
SCHEMBL28939454 0.83 RPS6KB1 (0.54) GPR119RPS6KB1AKT1MAP4K4
SCHEMBL19000161 0.81 GPR119 (0.52) GPR119NR1H2NR1H3EGLN2RET
SCHEMBL5128070 0.79 GPR119 (0.49) GPR119NR1H2NR1H3EGLN2MAP4K4
SCHEMBL21645241 0.77 GPR119 (0.37) GPR119RPS6KB1AKT1
SCHEMBL18980252 0.76 RPS6KB1 (0.48) RPS6KB1AKT1
SCHEMBL18980545 0.76 EIF2AK4 (0.42) RPS6KB1AKT1RETMAP4K4
SCHEMBL3922803 0.75 GPR119 (0.48) GPR119NR1H2NR1H3EGLN2RET
SCHEMBL26651056 0.75 GPR119 (0.44) GPR119NR1H2NR1H3EGLN2RET
SCHEMBL652792 0.75 GRM5 (0.53) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115485025-A Compounds and methods for modulating splicing 雷密克斯医疗公司 2022-12-16 CN disclosed