SCHEMBL28943005

SCHEMBL28943005

Nc1ccccc1NC(=O)c1ccc(F)c(N2C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 10/20 0.60
HDAC2 Q92769 7/20 0.50
HDAC3 O15379 6/20 0.50
PTGS1 P23219 2/20 0.50
MAPK1 P28482 1/20 0.50
HDAC4 P56524 3/20 0.49
HDAC7 Q8WUI4 3/20 0.49
HDAC10 Q969S8 2/20 0.49
HDAC11 Q96DB2 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
HDAC9 Q9UKV0 2/20 0.49
HDAC5 Q9UQL6 2/20 0.49
NCOR2 Q9Y618 1/20 0.49
NPSR1 Q6W5P4 1/20 0.48
GPR55 Q9Y2T6 1/20 0.48
MEN1 O00255 1/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
GRM1 Q13255 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28763802 0.87 HDAC1 (0.56) HDAC1HDAC2HDAC3MAPK1HDAC4
SCHEMBL28942997 0.86 HDAC1 (0.58) HDAC1HDAC2HDAC3PTGS1MAPK1
SCHEMBL29549466 0.80 POLB (0.62) HDAC1HDAC2HDAC3PTGS1MAPK1
SCHEMBL28763779 0.80 POLB (0.62) HDAC1HDAC2HDAC3PTGS1MAPK1
SCHEMBL29549870 0.77 ALDH1A1 (0.61) MEN1POLBKMT2ACA12
SCHEMBL28763787 0.77 ALDH1A1 (0.61) MEN1POLBKMT2ACA12
SCHEMBL4579192 0.75 HDAC2 (0.55) HDAC1HDAC2HDAC3NPSR1GPR55
SCHEMBL1063628 0.75 HDAC1 (1.00) HDAC1HDAC2HDAC3MAPK1HDAC4
SCHEMBL8401704 0.73 HDAC1 (0.89) HDAC1HDAC2HDAC3PTGS1MAPK1
SCHEMBL1065176 0.73 HDAC1 (0.78) HDAC1HDAC2HDAC3MAPK1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110452152-B 1, 3-dioxo isoindoline benzamide compound and application thereof 中国医学科学院药物研究所 2022-05-20 CN claimed
CN-110452152-B 1, 3-dioxo isoindoline benzamide compound and application thereof 中国医学科学院药物研究所 2022-05-20 CN disclosed