SCHEMBL28944232

SCHEMBL28944232

C[Si](C)(C)CCOCn1cc(-c2ccc(Nc3ccnc(N4Cc5ccc(S(C)(=O)=O)cc5C4)n3)cc2)cn1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 0.49
ROCK1 Q13464 4/20 0.48
HSP90AA1 P07900 5/20 0.38
HSP90AB1 P08238 5/20 0.38
FLT3 P36888 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637704 0.89 ROCK2 (0.65) ROCK2ROCK1
SCHEMBL29674785 0.78 ROCK2 (0.76) ROCK2ROCK1
SCHEMBL28777004 0.78 ROCK2 (0.76) ROCK2ROCK1
SCHEMBL24271321 0.75 KCNH2 (0.35) ROCK2ROCK1
SCHEMBL16637702 0.74 ROCK2 (0.44) ROCK2ROCK1
SCHEMBL28777011 0.72 ROCK2 (0.42) ROCK2ROCK1
SCHEMBL28777015 0.72 ROCK2 (0.42) ROCK2ROCK1
SCHEMBL29674607 0.72 ROCK2 (0.42) ROCK2ROCK1
SCHEMBL29674765 0.71 MAP4K4 (0.38)
SCHEMBL28777048 0.71 LCK (0.45) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114573566-B Selective ROCK2 kinase inhibitors 杭州邦顺制药有限公司 2023-05-30 CN disclosed
CN-114573566-A Selective ROCK2 kinase inhibitors 杭州邦顺制药有限公司 2022-06-03 CN disclosed