SCHEMBL28948857

SCHEMBL28948857

COc1ccccc1Cn1c(=O)[nH]c2c(N[C]=O)nc(-c3cccc(C(F)(F)F)c3)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 9/20 0.46
GRIN2B Q13224 9/20 0.46
THRB P10828 1/20 0.44
MTOR P42345 1/20 0.42
EPHX2 P34913 1/20 0.41
RXFP1 Q9HBX9 1/20 0.39
ADORA2A P29274 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90B1 P14625 1/20 0.39
TRAP1 Q12931 1/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28029213 0.89 ADORA2A (0.44) GRIN1GRIN2BMTOREPHX2ADORA2A
SCHEMBL28029238 0.87 MTOR (0.44) GRIN1GRIN2BMTORADORA2AMEN1
SCHEMBL28029224 0.87 MTOR (0.43) GRIN1GRIN2BMTORRXFP1ADORA2A
SCHEMBL28029222 0.87 CYP1A2 (0.54) GRIN1GRIN2BMTORADORA2AABCG2
SCHEMBL28028900 0.84 ADORA2A (0.46) MTOREPHX2ADORA2AMEN1USP2
SCHEMBL28198777 0.84 PIK3CA (0.44) MTORABCG2MEN1USP2LMNA
SCHEMBL28028874 0.84 MTOR (0.47) MTORADORA2AMEN1USP2LMNA
SCHEMBL28855796 0.83 MEN1 (0.41) GRIN1GRIN2BTHRBMTORADORA2A
SCHEMBL28028875 0.83 MTOR (0.42) GRIN1GRIN2BMTOREPHX2RXFP1
SCHEMBL28821952 0.83 MTOR (0.47) MTORADORA2AMEN1USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104870998-A Inhibition of phosphorylation of PRAS40, GSK 3-beta or P70S6K1 as a marker of TOR kinase inhibitory activity SIGNAL PHARM LLC 2015-08-26 CN disclosed