SCHEMBL289493

SCHEMBL289493

CC1(C(=O)O)CNC(=O)N1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AMPD2 Q01433 9/20 0.46
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.43
ELANE P08246 1/20 0.42
LMNA P02545 1/20 0.42
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3733166 0.76 TSHR (0.52) AMPD2ALDH1A1GAAELANELMNA
SCHEMBL7264096 0.73 HTR2C (0.47) ALDH1A1GAADDB1CRBNMEN1
SCHEMBL6001297 0.73 HTR2C (0.47) ALDH1A1GAADDB1CRBNMEN1
SCHEMBL15571839 0.72 ALDH1A1 (0.45) AMPD2ALDH1A1GAAELANELMNA
SCHEMBL2075062 0.72 ALDH1A1 (0.45) AMPD2ALDH1A1GAAELANELMNA
SCHEMBL6049149 0.72 ALDH1A1 (0.50) AMPD2ALDH1A1GAAELANELMNA
SCHEMBL13543074 0.70 KMT2A (0.48) ALDH1A1LMNADDB1CRBNGSK3A
SCHEMBL14664096 0.69 TSHR (0.48) AMPD2ALDH1A1LMNAKMT2A
SCHEMBL14828739 0.69 TSHR (0.51) AMPD2ALDH1A1GAALMNAKMT2A
SCHEMBL2246388 0.68 GAA (0.51) AMPD2ALDH1A1GAAELANELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427429-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS Abbott GmbH & Co. KG (DE) 2012-03-14 EP disclosed
WO-2010128102-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS ABBOTT GMBH & CO. KG (DE) 2010-11-11 WO disclosed